Biochemical interaction of anti-HCV telaprevir with the ABC transporters P-glycoprotein and breast cancer resistance protein

Table 4 IC ₅₀ values of telaprevir on [ ¹²⁵ I]-IAAP binding with P-gp or BCRP

	IC₅₀of telaprevir (μmol/L)
P-gp	16.5
BCRP	>80

ISSN: 1756-0500