Drug class | Compound | OL differentiationa | EC50, μM |
---|---|---|---|
SERM | Raloxifene | 82 | 0.1 |
Toremifene | 96 | 0.1 | |
Tamoxifen | 85 | 0.2 | |
Tricyclic anti-depressants | Perphenazine | 59 | 0.1 |
Fluphenazine | 91 | 0.1 | |
Prochlorperazine | 80 | 0.1 | |
Trifluoperazine | 60 | 0.2 | |
Quetiapine | 109 | 0.4 | |
Non-tricyclic anti-depressants | Perospirone | 88 | 0.1 |
Nitalapram | 51 | 1.1 | |
Escitalopram | 84 | 1.3 | |
Metylperon | 64 | 7.3 | |
Muscarinic | Benztropine | 66 | 0.3 |
Donepezil | 142 | 0.5 | |
Vesamicol | 91 | 1.4 | |
Oxybutynin | 67 | 2.6 | |
Ipatropium | 58 | 8.5 | |
Clemastineb | ND | 0.2 | |
Adrenergic | Salmeterol | 52 | 0.4 |
Betaxolol | 86 | 4.2 | |
Esmolol | 65 | 240 | |
Ion-channel | Ifenprodil | 93 | 0.4 |
Benproperine | 82 | 0.8 | |
Proxymetacaine | 77 | 1.0 | |
Dofetilide | 77 | 14 | |
DMPP | 97 | 13 | |
Anti-fungal | Bifonazole | 66 | 1.7 |